THE BEST SIDE OF LDN-27219 SIDE EFFECTS

1 especially intriguing compound is LDN-27219. Even though most tTG inhibitors are intended to bind towards the protein crosslinking Lively web-site, LDN-27219 in its place binds on the nucleotide binding pocket with the enzyme even though it is actually in its closed-state conformation, and stabilizes that conformation to circumvent crosslinking a